A-1155463 Robolid

A-1155463 RobolidA 1155463, a highly potent and selective BCL XL inhibitor, shows picomolar binding affinity to BCL XL, and >1000 fold weaker binding to BCL 2 and related proteins BCL W(Ki=19 nM) and MCL 1(Ki>440 nM).

BI-D1870 is an ATP-competitive inhibitor of S6 ribosome for RSK1/2/3/4 with IC50 of 31 nM/24 nM/18 nM/15 nM in cell-free assays

DTP3 is a selective GADD45

is an inhibitor of CDK9 and does not inhibit CDK2

2 nM and 0

Readability [d]: 10g

Fast and Precise Measurement

is an antineoplastic antimetabolite with immunosuppressant properties

Bisacodyl (INN) is a stimulant laxative drug that works directly on the colon to produce a bowel movement

acts on target cells in mammalian brain via stimulation of Histamine 1/2

less potent to Met

Acitretin is a second generation retinoid used for psoriasis

Internal adjustment